Publications in the Biomolecular Science and Medicinal Chemistry Division

Content: NG, V., KUEHNE, S. A. and CHAN, W.C., 2018. Rational design and synthesis of modified teixobactin analogues: in vitro antibacterial activity against Staphylococcus aureus, Propionibacterium acnes and Pseudomonas aeruginosa Chemistry - A European Journal. 24(36), 9136-9147

Content: CHAN, W.C., GENAPATHY, S. and YANG, L., 2018. Antibacterial compounds WO 2018/167506 A1 09/20/2018 00:00:00

Content: ZAMBERLAN, F., TURYANSKA, L., PATANE, A., LIU, Z., WILLIAMS, H. E. L., FAY, M. W., CLARKE, P. A., IMAMURA, Y., JIN, T., BRADSHAW, T. D., THOMAS, N. R. and GRABOWSKA, A. M., 2018. Stable DHLA-PEG capped PbS quantum dots: from synthesis to near-infrared biomedical imaging: Journal of Materials Chemistry B Journal of Materials Chemistry B. 6(4), 550-555

Content: BIN BREAK, MOHAMMED KHALED, HOSSAN, MD SHAHADAT, KHOO, YIVONN, QAZZAZ, MOHANNAD EMAD, AL-HAYALI, MOHAMMED Z. K., CHOW, SEK CHUEN, WIART, CHRISTOPHE, BRADSHAW, TRACEY D., COLLINS, HILARY and KHOO, TENG-JIN, 2018. Discovery of a highly active anticancer analogue of cardamonin that acts as an inducer of caspase-dependent apoptosis and modulator of the mTOR pathway FITOTERAPIA. 125, 161-173

Content: SANTOS, MARILIA S., NORTCLIFFE, ANDREW, LEWIS, WILLIAM, BRADSHAW, TRACEY D. and MOODY, CHRISTOPHER J., 2018. Synthesis of Highly Substituted 1,2-Diazetidin-3-ones, Small-Ring Scaffolds for Drug Discovery CHEMISTRY-A EUROPEAN JOURNAL. 24(33), 8325-+

Content: COUSIN, DAVID, HUMMERSONE, MARC G., BRADSHAW, TRACEY D., ZHANG, JIHONG, MOODY, CHRISTOPHER J., FOREITER, MAGDALENA B., SUMMERS, HELEN S., LEWIS, WILLIAM, WHEELHOUSE, RICHARD T. and STEVENS, MALCOLM F. G., 2018. Synthesis and growth-inhibitory activities of imidazo[5,1-d]-1,2,3,5-tetrazine-8-carboxamides related to the anti-tumour drug temozolomide, with appended silicon, benzyl and heteromethyl groups at the 3-position MEDCHEMCOMM. 9(3), 545-553

Content: CITOSSI, FRANCESCA, SMITH, THOMAS, LEE, JONG BONG, SEGAL, JOEL, GERSHKOVICH, PAVEL, STOCKS, MICHAEL J., BRADSHAW, TRACEY D., KELLAM, BARRIE and MARLOW, MARIA, 2018. Self-Assembling Benzothiazole-Based Gelators: A Mechanistic Understanding of in Vitro Bioactivation and Gelation MOLECULAR PHARMACEUTICS. 15(4), 1578-1586

Content: LEE JB, ZGAIR A, MALEC J, KIM TH, KIM MG, ALI J, QIN C, FENG W, CHIANG M, GAO X, VORONIN G, GARCES AE, LAU CL, CHAN TH, HUME A, MCINTOSH TM, SOUKARIEH F, AL-HAYALI M, CIPOLLA E, COLLINS HM, HEERY DM, SHIN BS, YOO SD, KAGAN L, STOCKS MJ, BRADSHAW TD, FISCHER PM and GERSHKOVICH P, 2018. Lipophilic activated ester prodrug approach for drug delivery to the intestinal lymphatic system. Journal of controlled release : official journal of the Controlled Release Society. 286, 10-19

Content: SMEDLEY, CHRISTOPHER J., STANLEY, PAUL A., QAZZAZ, MOHANNAD E., PROTA, ANDREA E., OLIERIC, NATACHA, COLLINS, HILARY, EASTMAN, HARRY, BARROW, ANDREW S., LIM, KUAN-HON, KAM, TOH-SEOK, SMITH, BRIAN J., DUIVENVOORDEN, HENDRIKA M., PARKER, BELINDA S., BRADSHAW, TRACEY D., STEINMETZ, MICHEL O. and MOSES, JOHN E., 2018. Sustainable Syntheses of (-)-Jerantinines A & E and Structural Characterisation of the Jerantinine-Tubulin Complex at the Colchicine Binding Site SCIENTIFIC REPORTS. 8,

Content: BLESSING ONYEGEME-OKERENTA, TRACEY BRADSHAW and KEITH SPRIGGS, 2018. Ethyl Acetate Extract of Senna alata (L) Roxb Increases Cytotoxicity in the Human Breast, Prostate and Colorectal Cancer Cells Journal of Cancer Treatment and Research. 6(3), 44-53

Content: BLESSING ONYEGEME-OKERENTA and TRACEY BRADSHAW, 2018. Anti-proliferative Activity of Ethyl Acetate Leaf Extract of Annona muricata L. on Selected Carcinoma Human Cell Lines London Journal of Research in Science: Natural and Formal. 18(4),

Content: BLESSING ONYEGEME-OKERENTA, CHRISTIAN AGYARE and TRACEY BRADSHAW, 2018. African Journal of Pharmacy and Pharmacology African Journal of Pharmacy and Pharmacology. 12(23), 310-318

Content: SKILLING, KATHRYN J., STOCKS, MICHAEL J., KELLAM, BARRIE, ASHFORD, MARIANNE, BRADSHAW, TRACEY D., BURROUGHS, LAURENCE and MARLOW, MARIA, 2018. Nucleoside-Based Self-Assembling Drugs for Localized Drug Delivery ChemMedChem. 13(11), 1098-1101

Content: PEREGO, PAOLA, HEMPEL, GEORG, LINDER, STIG, BRADSHAW, TRACEY D., LARSEN, ANNETTE K., PETERS, GODEFRIDUS J. and PHILLIPS, ROGER M., 2018. Cellular pharmacology studies of anticancer agents: recommendations from the EORTC-PAMM group CANCER CHEMOTHERAPY AND PHARMACOLOGY. 81(3), 427-441

Content: COUSIN, DAVID, HUMMERSONE, MARC, BRADSHAW, TRACEY D, ZHANG, JIHONG, MOODY, CHRISTOPHER J, FOREITER, MAGDALENA, SUMMERS, HELEN, LEWIS, WILLIAM, WHEELHOUSE, RT and STEVENS, MALCOLM FG, 2018. COD ID: 7121168 Crystallography Open Database.

Publications