Publications in the Biomolecular Science and Medicinal Chemistry Division

Content: BOUZINAB, KAOUTHAR, THOMAS, NEIL R., TURYANSKA, LYUDMILA, GERSHKOVICH, PAVEL, WESTON, NICOLA, ASHFORD, MARIANNE B. and BRADSHAW, TRACEY D., 2019. TARGETING BRAIN TUMOURS: APOFERRITIN NANOCAGE FOR DELIVERY OF NOVEL ANALOGUES OF TEMOZOLOMIDE NEURO-ONCOLOGY. 21, 4-4

Content: JC QUILLES, FR ROCHCO, CA MONTANARI, A LEITAO, VW MIGNONE, MA ARRUDA, L TURYANSKA and TD BRADSHAW, 2019. Apoferritin-encapsulation of cysteine protease inhibitors for cathepsin L inhibition in cancer cells. RSC Advances. 9, 36699-36706

Content: ABID, MOHAMMED, NOUCH, RYAN, BRADSHAW, TRACEY D., LEWIS, WILLIAM and WOODWARD, SIMON, 2019. Tripodal O-N-O Bis-Phenolato Amine Titanium(IV) Complexes Show High in vitro Anti-Cancer Activity EUROPEAN JOURNAL OF INORGANIC CHEMISTRY. 2774-2780

Content: YANG, ZHIKUAN, WEI, DANPING, DAI, XIAOLI, STEVENS, MALCOLM F. G., BRADSHAW, TRACEY D., LUO, YING and ZHANG, JIHONG, 2019. C8-Substituted Imidazotetrazine Analogs Overcome Temozolomide Resistance by Inducing DNA Adducts and DNA Damage FRONTIERS IN ONCOLOGY. 9,

Content: JISOOK LEE, NATALIE B. VINH, NYSSA DRINKWATER, WEI YANG, KOMAGAL KANNAN SIVARAMAN, LUKE S. SCHEMBRI, MICHELLE GAZDIK, PETER M. GRIN, GEORGINA S. BUTLER, CHRISTOPHER M. OVERALL, SUSAN A. CHARMAN, SHEENA MCGOWAN* and PETER J. SCAMMELLS*, 2019. Novel Human Aminopeptidase N Inhibitors: Discovery and Optimization of Subsite Binding Interactions Journal of Medicinal Chemistry. 62(15), 7185-7209

Content: LUKE S. SCHEMBRI, JONAS ERIKSSON and LUKE R. ODELL*, 2019. Palladium(0)-Catalyzed Carbonylative Synthesis of N-Acylsulfonamides via Regioselective Acylation The Journal of Organic Chemistry. 84(11), 6970-6981

Content: SANCHEZ J, LANE JR, CANALS M and STONE MJ, 2019. Influence of Chemokine N-Terminal Modification on Biased Agonism at the Chemokine Receptor CCR1. International journal of molecular sciences. 20(10),

Content: LEAVER DJ, CLEARY B, NGUYEN N, PRIEBBENOW DL, LAGIAKOS HR, SANCHEZ J, XUE L, HUANG F, SUN Y, MUJUMDAR P, MUDUDUDDLA R, VARGHESE S, TEGUH S, CHARMAN SA, WHITE KL, KATNENI K, CUELLAR M, STRASSER JM, DAHLIN JL, WALTERS MA, STREET IP, MONAHAN BJ, JARMAN KE, SABROUX HJ, FALK H, CHUNG MC, HERMANS SJ, PARKER MW, THOMAS T and BAELL JB, 2019. Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A. Journal of medicinal chemistry. 62(15), 7146-7159

Content: WARD SJ, GRATTON HE, INDRAYUDHA P, MICHAVILA C, MUKHOPADHYAY R, MAURER SK, CAULTON SG, EMSLEY J and DREVENY I, 2018. The structure of the deubiquitinase USP15 reveals a misaligned catalytic triad and an open ubiquitin-binding channel. The Journal of biological chemistry. 293(45), 17362-17374

Content: SALU BR, PANDO SC, BRITO MV, MEDINA AF, ODEI-ADDO F, FROST C, NAUDE R, SAMPAIO MU, EMSLEY J, MAFFEI FHA and OLIVA MLV, 2018. Improving the understanding of plasma kallikrein contribution to arterial thrombus formation using two plant protease inhibitors. Platelets. 30(3), 305-313

Content: PATHAK M, KAIRA BG, SLATER A and EMSLEY J, 2018. Cell Receptor and Cofactor Interactions of the Contact Activation System and Factor XI. Frontiers in medicine. 5, 66

Content: MOHAMMED BM, IVANOV I, MATAFONOV A, EMSLEY J and GAILANI D, 2018. Activity of Factor XII-Locarno. Research and practice in thrombosis and haemostasis. 2(1), 168-173

Content: LEE JB, ZGAIR A, MALEC J, KIM TH, KIM MG, ALI J, QIN C, FENG W, CHIANG M, GAO X, VORONIN G, GARCES AE, LAU CL, CHAN TH, HUME A, MCINTOSH TM, SOUKARIEH F, AL-HAYALI M, CIPOLLA E, COLLINS HM, HEERY DM, SHIN BS, YOO SD, KAGAN L, STOCKS MJ, BRADSHAW TD, FISCHER PM and GERSHKOVICH P, 2018. Lipophilic activated ester prodrug approach for drug delivery to the intestinal lymphatic system. Journal of controlled release : official journal of the Controlled Release Society. 286, 10-19

Content: LEK, NGEE, TADOKORO-CUCCARO, RIEKO, WHITCHURCH, JONATHAN B., MAZUMDER, BISMOY, MILES, HARRIET, PRENTICE, PHILIPPA, BUNCH, TREVOR, ZIELINSKA, KAROLINA, METZLER, VERONIKA, MONGAN, NIGEL P., HEERY, DAVID M. and HUGHES, IEUAN A., 2018. Predicting puberty in partial androgen insensitivity syndrome: Use of clinical and functional androgen receptor indices EBIOMEDICINE. 36, 401-409

Content: HEERY DM, 2018. A fellowship of Ring1 maintains AML stem cells. Blood. 131(16), 1771-1773

Publications